Publications

2021

Molecular Basis of Bicyclic Boronate β-Lactamase Inhibitors of Ultrabroad Efficacy – Insights From Molecular Dynamics Simulation Studies

E. Lence, C. González-Bello

Crambescin C1 Acts as A Possible Substrate of iNOS and eNOS Increasing Nitric Oxide Production and Inducing In Vivo Hypotensive Effect

J.A. Rubiolo, E. Lence, C. González-Bello, M. Roel, J. Gil-Longo, M. Campos-Toimil, E. Ternon, O.P. Thomas, A. González-Cantalapiedra, H. López-Alonso, M.R. Vieytes, L.M. Botana

6-Halopyridylmethylidene Penicillin-Based Sulfones Efficiently Inactivate the Natural Resistance of Pseudomonas aeruginosa to β-Lactam Antibiotics

J.C. Vázquez-Ucha, D. Rodríguez, C. Lasarte-Monterrubio, E. Lence, J. Arca-Suárez, M. Maneiro, E. Gato, A. Perez, M. Martínez-Guitián, C. Juan, A. Oliver, G. Bou, C. González-Bello, A. Beceiro

Bicyclic Boronate β‐Lactamase Inhibitors: The Present Hope against Deadly Bacterial Pathogens

E. Lence, C. González-Bello

Activity of imipenem, meropenem, cefepime, and sulbactam in combination with the β-lactamase inhibitor ln-1-255 against acinetobacter spp

C. Lasarte-Monterrubio, J.C. Vázquez-Ucha, M. Maneiro, J. Arca-Suárez, I. Alonso, P. Guijarro-Sánchez, J.D. Buynak, G. Bou, C. González-Bello, A. Beceiro

Molecular mechanisms driving in vivo development of OXA-10-mediated resistance to ceftolozane/tazobactam and ceftazidime/avibactam during treatment of extensively drug-resistant Pseudomonas aeruginosa infection

J. Arca-Suárez, C. Lasarte-Monterrubio, B.-K. Rodiño-Janeiro, G. Cabot, J. C. Vázquez-Ucha, P. M. Rodríguez-Iglesias, F. Galán-Sánchez, A. Beceiro, C. González-Bello, A. Oliver, G. Bou

2020

Characterization of the Locally Excited and Charge-transfer States of the Anticancer Drug Lapatinib by Ultrafast Spectroscopy and Computational Studies

I. Vayá, I.Andreu, E. Lence, C. González-Bello, M. C. Cuquerella, M. Navarrete-Miguel, D. Roca-Sanjuán, and M. A. Miranda

Protein Binding of Lapatinib and Its N- and O-Dealkylated Metabolites Interrogated by Fluorescence, Ultrafast Spectroscopy and Molecular Dynamics Simulations

I. Andreu, E. Lence, C. González-Bello, C. Mayorga, M.C. Cuquerella, I. Vaya, M.A. Miranda

Molecular and biochemical insights into the in vivo evolution of AmpC-mediated resistance to ceftolozane-tazobactam during treatment of a multidrug-resistant Pseudomonas aeruginosa infection 

J. Arca-Suárez, J.C. Vázquez-Ucha, P.A. Fraile-Ribot, E. Lence, G. Cabot, M. Martínez-Guitián, C. Lasarte-Monterrubio, M. Rodríguez-Iglesias, A. Beceiro, C. González-Bello, F. Galán-Sánchez, A. Oliver, G. Bou

Self‐Immolation of a Bacterial Dehydratase Enzyme by its Epoxide Product

E. Lence, M. Maneiro, M. Sanz-Gaitero, M.J. van Raaij, P. Thompson, A.R. Hawkins, C. González-Bello