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Publications

2012

Metal-assisted Ring-opening/closing Process of a Chiral Tetrahydroquinazoline
A. M. García-Deibe, J. Sanmartín-Matalobos, C. González-Bello, E. Lence, C. Portela-García, L. Martínez-Rodríguez, M. Fondo

Structural Variety of Zinc and Copper Complexes Based on a 2,3 Disubstituted 1,2,3,4-Tetrahydroquinazoline Ligand
J. Sanmartín Matalobos, C. Portela García, L. Martínez Rodríguez, C. González Bello, E. Lence, A.M. García-Deibe, M. Fondo

2011

A Prodrug Approach for Improving Antituberculosis Activity of Potent Mycobacterium tuberculosis Type II Dehydroquinase Inhibitors
L. Tizón, J. M. Otero, V. F. V. Prazeres, A. L. Llamas-Saiz, G. C. Fox, M. J. van Raaij, H. Lamb, A. R. Hawkins, J. M. Ainsa, L. Castedo, C. González-Bello

Tetrahydrobenzothiophene Derivatives as Inhibitors of type II Dehydroquinase
S. Paz, L. Tizón, J. M. Otero, A. L. Llamas-Saiz, G. C. Fox, M. J. van Raaij, H. Lamb, A. R. Hawkins, A. J. Lapthorn, L. Castedo, C. González-Bello

2010

Understanding the Key Factors that Control the Inhibition of Type 2 Dehydroquinase by (2R)-2-Benzyl-3-dehydroquinic acids
A. Peón, J. M. Otero, L. Tizón, V. F. V. Prazeres, A. L. Llamas-Saiz, G. C. Fox, M. J. Van Raaij, H. Lamb, A. R. Hawkins, F. Gago, L. Castedo, C. González-Bello

Synthesis and Biological Evaluation of New Nanomolar Competitive Inhibitors of Helicobacter pylori Type II Dehydroquinase. Structural Details of the Role of the Aromatic Moieties with Essential Residues
V. F. V. Prazeres, L. Tizón, J. M. Otero, P. Guardado-Calvo, A. L. Llamas-Saiz, M. J. van Raaij, L. Castedo, H. Lamb, A. R. Hawkins, C. González-Bello

Functional Desymmetrization of 1,3-Dioximes for the Obtention of 1,2,3-Hetero Trisubstituted Carbocycles
V. B. C. Figueira, A. G. Esqué, R. Varala, C.González-Bello, S. Prabhakar, A. M. Lobo

Tetrahedron Lett., 2010, 51, 2029-2031

Steady-State Fluorescence and Molecular Dynamic Studies on the Inhibition of Type II Dehydroquinase by (2R)-3-Benzyl-3-Dehydroquinic Acids
A. Peón, L. Tizón, V. F. V. Prazeres, L. Castedo, C. González-Bello

Drug of the Future, 2010, 35 (supl A), 175-176

Enol Mimics with a Flexible Side Chain as Inhibitors of Mycobacterium tuberculosis Dehydroquinase
B. Blanco, A. Sedes, C. Sánchez-Sixto, L. Castedo, C. González-Bello

Drug of the Future, 2010, 35 (supl A), 190

Competitive Inhibitors of Helicobacter Pylori Type II Dehydroquinase. Structural Details of the Role of the Aromatic Moieties Interactions with Essential Residues
V. F. V. Prazeres, L. Tizón, J. M. Otero, P. Guardado-Calvo, A. Llamas-Saiz, M. J. Van Raaij, L. Castedo, C. González-Bello

Drug of the Future, 2010, 35 (supl A), 190-191