Publicacións

2017

Structure-Based Rational Design of Adenosine Receptor Ligands

H. Gutiérrez-de-Terán, J. Sallander, E. Sotelo.

Multicomponent Assembly of the Kinesin Spindle Protein Inhibitor CPUYJ039 and Analogues as Antimitotic Agents

C. Carbajales, J. Sawada, G.i Marzaro, E. Sotelo, L. Escalante, A. Sánchez-Díaz Marta, X. García-Mera, A. Asai, A. Coelho

An efficient and recyclable 3D printed α-Al2O3 catalyst for the multicomponent assembly of bioactive heterocycles

J. Azuaje, C.R. Tubío, L. Escalante, M. Gómez, F. Guitián, A. Coelho, O. Caamaño, A. Gil, E. Sotelo

2016

Drug structural features affect drug delivery from hyperbranched polyesteramide hot melt extrudates

E. Raviña-Eirina, J. Azuaje, E. Sotelo, J. L. Gomez-Amoza, R. Martinez-Pacheco

Discovery of Potent and Highly Selective A2B Adenosine Receptor Antagonist Chemotypes

A. El Maatougui, J. Azuaje, M. González-Gómez, G. Miguez, A.Crespo, C. Carbajales, L. Escalante, X. García-Mera, H. Gutiérrez-de-Terán, E.Sotelo

3D printing of a heterogeneous copper-based catalyst

C. R. Tubío, J. Azuaje, L. Escalante, A. Coelho, F. Guitián, E. Sotelo, A. Gila.

2015

Pyrazin-2(1H)-ones as a novel class of selective A3 adenosine receptor antagonists

J. Azuaje, C. Carbajales, M. González Gómez, A. Coelho, O. Caamaño, H. Gutiérrez de Terán, E. Sotelo

Integrated Ugi-Based Assembly of Functionally, Skeletally, and Stereochemically Diverse 1,4-Benzodiazepin-2-ones

J. Azuaje, J. M. Pérez.Rubio, V. Yaziji, A. El Maatougui, J. C. González.Gomez, V. M. Sánchez.Pedregal, A. Navarro.Vázquez, C. F. Masaguer, M. Teijeira, E. Sotelo

Sol–gel entrapped Cu in a silica matrix: An efficient heterogeneous nanocatalyst for Huisgen and Ullmann intramolecular coupling reactions

P. Diz, P. Pernas,, A. El Maatougui, C. R. Tubio, J. Azuaje, E. Sotelo, F. Guitián, A. Gil, Al. Coelho

Multicomponent Reactions in Antimitotic Drug Discovery

A. Cores, C. Carbajales, A. Coelho